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PF-04531083

Chemical Structure : PF-04531083

CAS No.: 1079400-07-9

PF-04531083 (PF-4531083, PF 04531083)

Catalog No.: PC-61870Not For Human Use, Lab Use Only.

PF-04531083 (PF 4531083) is a potent and selective, orally available sodium channel Nav1.8 blocker for treatment of pain.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

PF-04531083 (PF 4531083) is a potent and selective, orally available sodium channel Nav1.8 blocker for treatment of pain.

Physicochemical Properties

M.Wt 357.798
Formula C17H16ClN5O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

N-[6-amino-5-(2-chloro-5-methoxyphenyl)pyridin-2-yl]-2-methylpyrazole-3-carboxamide

References

1. Bagal SK, et al. Bioorg Med Chem Lett. 2014 Aug 15;24(16):3690-9.

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