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PF-04958242

Chemical Structure : PF-04958242

CAS No.: 1258963-59-5

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PF-04958242 (Pesampator, PF04958242)

Catalog No.: PC-61864Not For Human Use, Lab Use Only.

PF-04958242 (Pesampator) is a novel potent, selctive, and orally-active AMPA receptor (AMPAR) positive allosteric modulator (PAM) with Ki of 170 nM, EC50 of 370 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

PF-04958242 (Pesampator) is a novel potent, selctive, and orally-active AMPA receptor (AMPAR) positive allosteric modulator (PAM) with Ki of 170 nM, EC50 of 370 nM.
PF-04958242 (Pesampator) is under development for the treatment of cognitive symptoms in schizophrenia.

Physicochemical Properties

M.Wt 392.49
Formula C18H20N2O4S2
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

N-((3S,4S)-4-(4-(5-cyano-2-thienyl)phenoxy)tetrahydro-3-furanyl)-2-propanesulfonamide

References

1. Shaffer CL, et al. J Med Chem. 2015 May 28;58(10):4291-308.

2. Ranganathan M, et al. Mol Psychiatry. 2017 Feb 28. doi: 10.1038/mp.2017.6.

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