PF-05150122 |CAS:1235406-03-7 Probechem Biochemicals

Chemical Structure : PF-05150122

CAS No.: 1235406-03-7

Catalog No.: PC-63176Not For Human Use, Lab Use Only.

PF-05150122 is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 21 nM, no significant activity against Nav1.5.

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Biological Activity

PF-05150122 is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 21 nM, no significant activity against Nav1.5.

M.Wt	531.885
Formula	C19H10ClF4N5O3S2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	5-chloro-2-fluoro-4-(2-(pyridazin-4-yl)-4-(trifluoromethyl)phenoxy)-N-(1,3,4-thiadiazol-2-yl)benzenesulfonamide

1. Swain NA, et al. J Med Chem. 2017 Aug 24;60(16):7029-7042.

2. Jones HM, et al. Clin Pharmacokinet. 2016 Jul;55(7):875-87.