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Chemical Structure : PF-05150122
CAS No.: 1235406-03-7
Catalog No.: PC-63176Not For Human Use, Lab Use Only.
PF-05150122 is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 21 nM, no significant activity against Nav1.5.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $258 | In stock | |
| 10 mg | $398 | In stock | |
| 50 mg | Get quote | ||
| 100 mg | Get quote |
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PF-05150122 is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 21 nM, no significant activity against Nav1.5.
| M.Wt | 531.885 | |
| Formula | C19H10ClF4N5O3S2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
5-chloro-2-fluoro-4-(2-(pyridazin-4-yl)-4-(trifluoromethyl)phenoxy)-N-(1,3,4-thiadiazol-2-yl)benzenesulfonamide |
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1. Swain NA, et al. J Med Chem. 2017 Aug 24;60(16):7029-7042.
2. Jones HM, et al. Clin Pharmacokinet. 2016 Jul;55(7):875-87.
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