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PF-05212377

Chemical Structure : PF-05212377

CAS No.: 1226793-34-5

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PF-05212377 (SAM-760;PF 5212377)

Catalog No.: PC-35004Not For Human Use, Lab Use Only.

PF-05212377 (SAM-760, PF 5212377) is a potent and selective 5-HT6 receptor antagonist with Ki of 0.32 nM (human 5HT6), shows potential therapy for the symptomatic treatment of mild to moderate Alzheimer's disease.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    PF-05212377 (SAM-760, PF 5212377) is a potent and selective 5-HT6 receptor antagonist with Ki of 0.32 nM (human 5HT6), shows potential therapy for the symptomatic treatment of mild to moderate Alzheimer's disease.

    Physicochemical Properties

    M.Wt 356.444
    Formula C18H20N4O2S
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    2-methyl-1-(phenylsulfonyl)-4-(piperazin-1-yl)-1H-benzo[d]imidazole

    References

    1. Fullerton T, et al. Alzheimers Res Ther. 2018 Apr 5;10(1):38.

    2. Fullerton T, et al. Alzheimers Res Ther. 2018 Apr 5;10(1):38.

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