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PF-05661014

Chemical Structure : PF-05661014

CAS No.: 2153474-85-0

PF-05661014 (PF05661014)

Catalog No.: PC-35155Not For Human Use, Lab Use Only.

PF-05661014 is a potent, selective Nav1.3 inhibitor with IC50 of 0.26 uM, shows no activity for Nav1.7 (IC50>10 uM).

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

PF-05661014 is a potent, selective Nav1.3 inhibitor with IC50 of 0.26 uM, shows no activity for Nav1.7 (IC50>10 uM).

Physicochemical Properties

M.Wt 388.46
Formula C17H16N4O3S2
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

4-(3-benzylureido)-N-(thiazol-2-yl)benzenesulfonamide

References

1. Wang L, et al. Br J Pharmacol. 2015 Oct;172(20):4905-18.

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