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PF-4181366

Chemical Structure : PF-4181366

CAS No.: 1082743-32-5

PF-4181366 (PF-04181366, PF04181366, PF4181366)

Catalog No.: PC-60206Not For Human Use, Lab Use Only.

PF-4181366 (PF-04181366) is a potent, selective, brain penetrant PDE9A inhibitor with IC50 of 1.8 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    PF-4181366 (PF-04181366) is a potent, selective, brain penetrant PDE9A inhibitor with IC50 of 1.8 nM.
    PF-4181366 (PF-04181366) displays >25-fold selectivity over other PDEs.

    Physicochemical Properties

    M.Wt 429.53
    Formula C24H27N7O
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    4H-Pyrazolo(3,4-d)pyrimidin-4-one, 1-cyclopentyl-1,5-dihydro-6-((3S,4S)-4-methyl-1-(6-quinoxalinylmethyl)-3-pyrrolidinyl)-

    References

    1. Verhoest PR, et al. J Med Chem. 2009 Dec 24;52(24):7946-9.

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