PI3K inhibitor X (Pilaralisib analogue) | class I PI3K inhibitor

Chemical Structure : PI3K inhibitor X

CAS No.: 956958-53-5

PI3K inhibitor X (XL147 analog, Pilaralisib analogue)

Catalog No.: PC-42812Not For Human Use, Lab Use Only.

PI3K inhibitor X (XL-147 analog) is a derivative of XL147 that acts as a reversible inhibitor of class I PI3Ks with IC50 of 39, 36, 23 and 383 nM for p110α, δ, γ and β respectively.

Packing	Price	Stock
10 mg	$88	In stock
25 mg	$148	In stock
50 mg	$258	In stock
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Biological Activity

PI3K inhibitor X (XL147 analog) is a derivative of XL147 that acts as a reversible inhibitor of class I PI3Ks with IC50 of 39, 36, 23 and 383 nM for p110α, δ, γ and β respectively.
Compound 147 in patent WO2012006552A1.

Physicochemical Properties

M.Wt	448.5208
Formula	C21H16N6O2S2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	Benzenesulfonamide, N-[3-(2,1,3-benzothiadiazol-5-ylamino)-2-quinoxalinyl]-4-methyl-

References

1. Carlos L. Arteaga, et al. Combinations of kinase inhibitors for the treatment of cancer. WO 2012006552 A1.

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PI3K inhibitor X (XL147 analog, Pilaralisib analogue)

Biological Activity

Physicochemical Properties

References

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