PITCOIN4

Chemical Structure : PITCOIN4

Catalog No.: PC-23002Not For Human Use, Lab Use Only.

PITCOIN4 is a potent, highly selective inhibitor of class II alpha PI3K (PI3K-C2α) with IC50 of 56 nM, >100-fold selectivity over PI3K-C2β.

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Biological Activity

PITCOIN4 is a potent, highly selective inhibitor of class II alpha PI3K (PI3K-C2α) with IC50 of 56 nM, >100-fold selectivity over PI3K-C2β.

M.Wt	599.73
Formula	C30H29N7O3S2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(4-(2-oxo-2-((2-phenylpropan-2-yl)amino)ethyl)thiazol-2-yl)-2-((4-oxo-3-phenethyl-3,4-dihydropteridin-2-yl)thio)acetamide

1. Murat Kücükdisli, et al. J Med Chem. 2023 Oct 26;66(20):14278-14302.