PSB-SB-487 | GPR55 inhibitor | Probechem Biochemicals

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Chemical Structure : PSB-SB-487

CAS No.: 1399049-81-0

PSB-SB-487 (GPR55 antagonist)

Catalog No.: PC-38506Not For Human Use, Lab Use Only.

PSB-SB-487 is a potent, selective antagonist of orphan G-protein-coupled receptor GPR55 with IC50 value 113 nM, and KB value 561 nM (hGPR55), shows little to no activity against CB1/CB2 and GPR18 receptors.

Packing	Price	Stock
5 mg	$138	In stock
10 mg	$218	In stock
25 mg	$378	In stock
50 mg	$598	In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

PSB-SB-487 is a potent, selective antagonist of orphan G-protein-coupled receptor GPR55 with IC50 value 113 nM, and KB value 561 nM (hGPR55), shows little to no activity against CB1/CB2 and GPR18 receptors.

Physicochemical Properties

M.Wt	408.538
Formula	C26H32O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	5-hydroxy-3-(2-hydroxybenzyl)-7-(2-methylnonan-2-yl)-2H-chromen-2-one

References

1. Viktor Rempel, et al. J Med Chem. 2013 Jun 13;56(11):4798-810.

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PSB-SB-487 (GPR55 antagonist)

Biological Activity

Physicochemical Properties

References

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