Pirenzepine | M1 mAChR antagonist | Probechem Biochemicals

Chemical Structure : Pirenzepine

CAS No.: 28797-61-7

Pirenzepine (LS 519, Pirenzepin, Gastrozepin)

Catalog No.: PC-23330Not For Human Use, Lab Use Only.

Pirenzepine (LS519, Pirenzepin, Gastrozepin) is a selective M1 mAChR (muscarinic acetylcholine receptor) antagonist, shows gastric secretion-inhibitory action but without central-nervous sedation.

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Biological Activity

Pirenzepine (LS519, Pirenzepin, Gastrozepin) is a selective M1 mAChR (muscarinic acetylcholine receptor) antagonist, shows gastric secretion-inhibitory action but without central-nervous sedation.

Physicochemical Properties

M.Wt	351.41
Formula	C19H21N5O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	11-(2-(4-Methylpiperazin-1-yl)acetyl)-5,11-dihydro-6H-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one

References

1. Eberlein W, et al. Arzneimittelforschung. 1977 Feb;27(2):356-9.

2. Brunner H, et al. Arzneimittelforschung. 1977;27(3):684-7.

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Pirenzepine (LS 519, Pirenzepin, Gastrozepin)

Biological Activity

Physicochemical Properties

References

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