Welcome to ProbeChem!Global Supplier of Chemical Probes, Inhibitors & Agonists.
Chemical Structure : Pitolisant
CAS No.: 362665-56-3
Catalog No.: PC-42909Not For Human Use, Lab Use Only.
Pitolisant (Tiprolisant, BF-2649, BF 2.649) is a potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $78 | In stock | |
| 25 mg | $138 | In stock | |
| 50 mg | $218 | In stock | |
| 100 mg | $358 | In stock | |
| 250 mg | Get quote |
Bulk size, bulk discount!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
Pitolisant (Tiprolisant, BF-2649, BF 2.649) is a potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM.
Pitolisant shows no effect on H1, H2, H4 receptors (IC50>10 uM).
Pitolisant is orally bioactive.
| M.Wt | 295.8474 | |
| Formula | C17H26ClNO | |
| Appearance | Solid | |
| Storage |
|
|
| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
Piperidine, 1-[3-[3-(4-chlorophenyl)propoxy]propyl]- |
|
1. Ligneau X, et al. J Pharmacol Exp Ther. 2007 Jan;320(1):365-75.
2. Dudek M, et al. Metab Brain Dis. 2016 Oct;31(5):1023-9.
3. Ligneau X, et al. Biochem Pharmacol. 2007 Apr 15;73(8):1215-24.
Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright
