Pitolisant oxalate |CAS:362665-57-4 Probechem Biochemicals

Chemical Structure : Pitolisant oxalate

CAS No.: 362665-57-4

Catalog No.: PC-42910Not For Human Use, Lab Use Only.

A potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

A potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM; no effect on H1, H2, H4 receptors (IC50>10 uM); orally bioactive.

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Approved

M.Wt	385.8823
Formula	C19H28ClNO5
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Piperidine, 1-[3-[3-(4-chlorophenyl)propoxy]propyl]-, ethanedioate (1:1)

1. Ligneau X, et al. J Pharmacol Exp Ther. 2007 Jan;320(1):365-75.

2. Dudek M, et al. Metab Brain Dis. 2016 Oct;31(5):1023-9.

3. Ligneau X, et al. Biochem Pharmacol. 2007 Apr 15;73(8):1215-24.