Pyk2-IN-25a |CAS:2052970-45-1 Probechem Biochemicals

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Chemical Structure : Pyk2-IN-25a

Pyk2-IN-25a

Catalog No.: PC-62798Not For Human Use, Lab Use Only.

Pyk2-IN-25a is a highly potent Pyk2 (PTK2B) inhibitor with IC50 of 0.67 nM, dispalys 2-fold weakening potency for FAK (IC50=1.26 nM).

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Pyk2-IN-25a is a highly potent Pyk2 (PTK2B) inhibitor with IC50 of 0.67 nM, dispalys 2-fold weakening potency for FAK (IC50=1.26 nM).
Pyk2-IN-25a is a suitable tool compound for future proof-of-concept studies.

Physicochemical Properties

M.Wt	478.494
Formula	C21H21F3N6O2S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	7-(methylsulfonyl)-35-(trifluoromethyl)-2,4,7-triaza-3(2,4)-pyrimidina-6(3,2)-pyridina-1(1,3)-benzenacyclodecaphane

References

1. Farand J, et al. Bioorg Med Chem Lett. 2016 Dec 15;26(24):5926-5930.

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Pyk2-IN-25a

Biological Activity

Physicochemical Properties

References

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