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Pyk2-IN-25a

Chemical Structure : Pyk2-IN-25a

CAS No.: 2052970-45-1

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Pyk2-IN-25a

Catalog No.: PC-62798Not For Human Use, Lab Use Only.

Pyk2-IN-25a is a highly potent Pyk2 (PTK2B) inhibitor with IC50 of 0.67 nM, dispalys 2-fold weakening potency for FAK (IC50=1.26 nM).

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    Pyk2-IN-25a is a highly potent Pyk2 (PTK2B) inhibitor with IC50 of 0.67 nM, dispalys 2-fold weakening potency for FAK (IC50=1.26 nM).
    Pyk2-IN-25a is a suitable tool compound for future proof-of-concept studies.

    Physicochemical Properties

    M.Wt 478.494
    Formula C21H21F3N6O2S
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    7-(methylsulfonyl)-35-(trifluoromethyl)-2,4,7-triaza-3(2,4)-pyrimidina-6(3,2)-pyridina-1(1,3)-benzenacyclodecaphane

    References

    1. Farand J, et al. Bioorg Med Chem Lett. 2016 Dec 15;26(24):5926-5930.

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