R995045 | Delta Opioid agonist | Probechem Biochemicals

Chemical Structure : R995045

R995045 (R 995045, R-995045)

Catalog No.: PC-72734Not For Human Use, Lab Use Only.

R995045 is a novel δ-opioid receptor (δOR) agonist with pKi of 5.94, cAMP pIC50 of 6.01, >10-fold selectivity over µOR and κOR.

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Biological Activity

R995045 is a novel δ-opioid receptor (δOR) agonist with pKi of 5.94, cAMP pIC50 of 6.01, >10-fold selectivity over µOR and κOR.
R995045 acts as a negative allosteric modulator for leu-enkephalin potency in the cAMP glosensor assay.

Physicochemical Properties

M.Wt	342.373
Formula	C16H14N4O3S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N'-(2-hydroxy-3-methoxybenzylidene)-3-(2-thienyl)-1H-pyrazole-5-carbohydrazide

References

1. Meqbil YJ, et al. Molecules. 2021 Nov 29;26(23):7236.

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R995045 (R 995045, R-995045)

Biological Activity

Physicochemical Properties

References

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