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Chemical Structure : R995045
Catalog No.: PC-72734Not For Human Use, Lab Use Only.
R995045 is a novel δ-opioid receptor (δOR) agonist with pKi of 5.94, cAMP pIC50 of 6.01, >10-fold selectivity over µOR and κOR.
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R995045 is a novel δ-opioid receptor (δOR) agonist with pKi of 5.94, cAMP pIC50 of 6.01, >10-fold selectivity over µOR and κOR.
R995045 acts as a negative allosteric modulator for leu-enkephalin potency in the cAMP glosensor assay.
| M.Wt | 342.373 | |
| Formula | C16H14N4O3S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Meqbil YJ, et al. Molecules. 2021 Nov 29;26(23):7236.
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