RU-TRAAK-2

Chemical Structure : RU-TRAAK-2

CAS No.: 1210538-56-9

Catalog No.: PC-70312Not For Human Use, Lab Use Only.

RU-TRAAK-2 is a completely reversible K2P channel TRAAK (KCNK4, K2P4.1) inhibitor with IC50 of 0.719 uM for TRAAK-mediated efflux, shows no activity for non-K2P channels (Kv1.2, Slo1 and GIRK2).

Packing	Price	Stock
5 mg	$98	In stock
10 mg	$148	In stock
25 mg	$258	In stock
50 mg		Get quote
100 mg		Get quote

Get Quotation Now

* Please select Quantity before adding items.

or Bulk Inquiry

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Biological Activity

RU-TRAAK-2 is a completely reversible K2P channel TRAAK (KCNK4, K2P4.1) inhibitor with IC50 of 0.719 uM for TRAAK-mediated efflux, shows no activity for non-K2P channels (Kv1.2, Slo1 and GIRK2).

Physicochemical Properties

M.Wt	335.425
Formula	C19H17N3OS
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1-(benzo[d]thiazol-2-ylmethyl)-1-methyl-3-(3-phenylprop-2-yn-1-yl)urea

References

1. Su Z, et al. Proc Natl Acad Sci U S A. 2016 May 17;113(20):5748-53.

2. Cancer Res. 2017 Aug 15;77(16):4293-4304.

Overnight Delivery
Fast & Safe Delivery Worldwide
Rewards Program

About Us

Our Services

Site Map

Join with Us
Product Use Citations

Pharmacological Glossary Abbreviations

Abbreviations

Quality Manual

Inquiry Form
How to Order

Terms & Conditions

Credit Card Payment

Shipping Rates & Policies

Privacy Policy
sales@probechem.com

RU-TRAAK-2

Biological Activity

Physicochemical Properties

References

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

Get Quote

* Indicates a Required FieldYour information is safe with us.