Radiprodil | GluN2B antagonist | Probechem Biochemicals

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Chemical Structure : Radiprodil

CAS No.: 496054-87-6

Radiprodil (RGH-896, RGH896)

Catalog No.: PC-25808Not For Human Use, Lab Use Only.

Radiprodil (RGH-896) is a selective, negative allosteric modulator / antagonist of GluN2B-containing NMDA receptors (GluN2B) with IC50 of 3-10 nM, with no activity against NR2A receptors.

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5 mg	$88	In stock
10 mg	$128	In stock
25 mg	$218	In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Radiprodil (RGH-896) is a selective, negative allosteric modulator / antagonist of GluN2B-containing NMDA receptors (GluN2B) with IC50 of 3-10 nM, with no activity against NR2A receptors.

Physicochemical Properties

M.Wt	397.41
Formula	C21H20FN3O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	2-(4-(4-Fluorobenzyl)piperidin-1-yl)-2-oxo-N-(2-oxo-2,3-dihydrobenzo[d]oxazol-6-yl)acetamide

References

1. Bertocchi I, et al. Br J Pharmacol. 2024 Jun;181(12):1886-1894.

2. Michel A, et al. PLoS One. 2015 Aug 31;10(8):e0135949.

3. Rammes G, et al. Neuropharmacology. 2018 Sep 15;140:184-192.

4. Romain Labas, et al. Eur J Med Chem. 2011 Jun;46(6):2295-309.

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Radiprodil (RGH-896, RGH896)

Biological Activity

Physicochemical Properties

References

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