Chemical Structure : Ralaniten
CAS No.: 1203490-23-6
Catalog No.: PC-60529Not For Human Use, Lab Use Only.
Ralaniten (EPI-002) is a novel small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor, inhibits AR transcriptional activity with IC50 of 7.4 uM.
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Ralaniten (EPI-002) is a novel small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor, inhibits AR transcriptional activity with IC50 of 7.4 uM.
AR NTD-targeting agents have the potential to overcome shortcomings of current hormonal therapies by inhibiting all forms of AR-mediated transcriptional activity, and as a result, may affect a broader AR population including mutational and splice variant ARs.
M.Wt | 394.89 | |
Formula | C21H27ClO5 | |
Appearance | Solid | |
Storage |
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Solubility |
10 mM in DMSO |
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Chemical Name/SMILES |
(2R)-3-[4-(2-{4-[(2S)-3-chloro- 2-hydroxypropoxy]phenyl}propan-2-yl)phenoxy]propane- 1,2-diol |
1. Antonarakis ES, et al. Oncologist. 2016 Dec;21(12):1427-1435.
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