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Chemical Structure : Relebactam
CAS No.: 1174018-99-5
Catalog No.: PC-45070Not For Human Use, Lab Use Only.
Relebactam (MK-7655) is a novel β-lactamase inhibitor that inhibited both class A and C β-lactamases in vitro.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $105 | In stock | |
| 25 mg | $345 | In stock | |
| 100 mg | $785 | In stock | |
| 500 mg | Get quote |
Bulk size, bulk discount!
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Relebactam (MK-7655) is a novel β-lactamase inhibitor that inhibited both class A and C β-lactamases in vitro; effectively restored imipenem's activity against imipenem-resistant Pseudomonas and Klebsiella strains at clinically achievable concentrations; reduces imipenem MICs for Enterobacteriaceae with KPC carbapenemases from 16-64 mg/L to 0.12-1 mg/L at a concentration of 4 mg/L.
Bacterial Infection
Phase 3 Clinical
| M.Wt | 348.3754 | |
| Formula | C12H20N4O6S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
Sulfuric acid, mono[(1R,2S,5R)-7-oxo-2-[(4-piperidinylamino)carbonyl]-1,6-diazabicyclo[3.2.1]oct-6-yl] ester |
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1. Hirsch EB, et al. Antimicrob Agents Chemother. 2012 Jul;56(7):3753-7.
2. Blizzard TA, et al. Bioorg Med Chem Lett. 2014 Feb 1;24(3):780-5.
3. Livermore DM, et al. J Antimicrob Chemother. 2013 Oct;68(10):2286-90.
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