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Relebactam

Chemical Structure : Relebactam

CAS No.: 1174018-99-5

Relebactam (MK-7655, MK7655)

Catalog No.: PC-45070Not For Human Use, Lab Use Only.

Relebactam (MK-7655) is a novel β-lactamase inhibitor that inhibited both class A and C β-lactamases in vitro.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Relebactam (MK-7655) is a novel β-lactamase inhibitor that inhibited both class A and C β-lactamases in vitro.
Relebactam (MK-7655) effectively restored imipenem's activity against imipenem-resistant Pseudomonas and Klebsiella strains at clinically achievable concentrations.
Relebactam (MK-7655) reduces imipenem MICs for Enterobacteriaceae with KPC carbapenemases from 16-64 mg/L to 0.12-1 mg/L at a concentration of 4 mg/L.

Physicochemical Properties

M.Wt 348.3754
Formula C12H20N4O6S
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

Sulfuric acid, mono[(1R,2S,5R)-7-oxo-2-[(4-piperidinylamino)carbonyl]-1,6-diazabicyclo[3.2.1]oct-6-yl] ester

References

1. Hirsch EB, et al. Antimicrob Agents Chemother. 2012 Jul;56(7):3753-7.

2. Blizzard TA, et al. Bioorg Med Chem Lett. 2014 Feb 1;24(3):780-5.

3. Livermore DM, et al. J Antimicrob Chemother. 2013 Oct;68(10):2286-90.

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