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Rilmenidine

Chemical Structure : Rilmenidine

CAS No.: 54187-04-1

Rilmenidine

Catalog No.: PC-23251Not For Human Use, Lab Use Only.

Rilmenidine is a potent, selective and orally active I1 imidazoline receptor (I1R) agonist with 83.1 nM, displays some selectivity for I1Rs over α2ARs, shows antihypertensive effect.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

Rilmenidine is a potent, selective and orally active I1 imidazoline receptor (I1R) agonist with 83.1 nM, displays some selectivity for I1Rs over α2ARs, shows antihypertensive effect.

Physicochemical Properties

M.Wt 180.25
Formula C10H16N2O
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

N-(Dicyclopropylmethyl)-4,5-dihydrooxazol-2-amine

References

1. Gasparik V, et al. J Med Chem. 2015 Jan 22;58(2):878-87.

2. Reid JL. Rilmenidine: a clinical overview. Am J Hypertens. 2000;13(6 Pt 2):106S-111S.

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