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SAS-1121

Chemical Structure : SAS-1121

CAS No.: 2095551-67-8

SAS-1121 (SAS 1121;SAS1121)

Catalog No.: PC-61103Not For Human Use, Lab Use Only.

SAS-1121 is a novel potent, subtype-selective sigma 2 receptor/PGRMC1 ligand with Ki of 16.2 nM, 574-fold selectivity over sigma 1 receptors.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    SAS-1121 is a novel potent, subtype-selective sigma 2 receptor/PGRMC1 ligand with Ki of 16.2 nM, 574-fold selectivity over sigma 1 receptors.

    Physicochemical Properties

    M.Wt 477.605
    Formula C28H35N3O4
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    benzyl (1R,5S)-8-(4-(3-ethoxy-3-oxopropyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine-2-carboxylate

    References

    1. Sahn JJ, et al. ChemMedChem. 2016 Mar 17;11(6):556-61.

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