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SB-699551

Chemical Structure : SB-699551

CAS No.: 791789-61-2

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SB-699551 (SB699551)

Catalog No.: PC-38716Not For Human Use, Lab Use Only.

SB699551 is a potent, selective 5-HT5A receptor antagonist with pKi of 8.3, >100-fold selectivity over 5-HT1B/D, 5-HT2A, 5-HT2C, 5-HT1A and 5-HT7 receptors.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

SB699551 is a potent, selective 5-HT5A receptor antagonist with pKi of 8.3, >100-fold selectivity over 5-HT1B/D, 5-HT2A, 5-HT2C, 5-HT1A and 5-HT7 receptors.
SB699551 also is a novel PSMD4/Rpn10 inhibitor, decreases cell viability in MM cell lines.

Physicochemical Properties

M.Wt 511.754
Formula C34H45N3O
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

N-[2-(Dimethylamino)ethyl]-N-[[4'-[[(2-phenylethyl)amino]methyl][1,1'-biphenyl]-4-yl]methyl]cyclopentanepropanamide

References

1. Thomas DR, et al. Neuropharmacology. 2006 Sep;51(3):566-77.

2. Du T, et al. Blood. 2023 Jan 11:blood.2022017897.

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