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Chemical Structure : SB 204741
CAS No.: 152239-46-8
Catalog No.: PC-38060Not For Human Use, Lab Use Only.
SB 204741 is a potent and selective 5-HT2B receptor antagonist (pA2=7.95).
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|---|---|---|---|
| 5 mg | $148 | In stock | |
| 10 mg | $238 | In stock | |
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| 100 mg | Get quote |
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SB 204741 is a potent and selective 5-HT2B receptor antagonist (pA2=7.95).
SB 204741 displays >135-fold selectivity over 5-HT2C (pKi =5.82), 5-HT2A (pKi <5.2), 5-HT1A, 1D, 1E, 5-HT3 and 5-HT4 receptors.
| M.Wt | 286.35 | |
| Formula | C14H14N4OS | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
N-(1-Methyl-1H-indolyl-5-yl)-N''-(3-methyl-5-isothiazolyl)urea |
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1. Bonhaus DW, et al. Br J Pharmacol. 1995 Jun;115(4):622-8.
2. Prins NH, et al. Br J Pharmacol. 1997 Feb;120(4):714-20.
3. Glusa E, et al. Br J Pharmacol. 2000 Jun;130(3):692-8.
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