SB 204741 |CAS:152239-46-8 Probechem Biochemicals

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Chemical Structure : SB 204741

CAS No.: 152239-46-8

SB 204741 (SB204741)

Catalog No.: PC-38060Not For Human Use, Lab Use Only.

SB 204741 is a potent and selective 5-HT2B receptor antagonist (pA2=7.95).

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5 mg	$148	In stock
10 mg	$238	In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

SB 204741 is a potent and selective 5-HT2B receptor antagonist (pA2=7.95).
SB 204741 displays >135-fold selectivity over 5-HT2C (pKi =5.82), 5-HT2A (pKi <5.2), 5-HT1A, 1D, 1E, 5-HT3 and 5-HT4 receptors.

Physicochemical Properties

M.Wt	286.35
Formula	C14H14N4OS
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(1-Methyl-1H-indolyl-5-yl)-N''-(3-methyl-5-isothiazolyl)urea

References

1. Bonhaus DW, et al. Br J Pharmacol. 1995 Jun;115(4):622-8.

2. Prins NH, et al. Br J Pharmacol. 1997 Feb;120(4):714-20.

3. Glusa E, et al. Br J Pharmacol. 2000 Jun;130(3):692-8.

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SB 204741 (SB204741)

Biological Activity

Physicochemical Properties

References

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