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SCO-240

Chemical Structure : SCO-240

CAS No.: 1695564-98-7

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SCO-240 (SCO240, SCO 240)

Catalog No.: PC-26763Not For Human Use, Lab Use Only.

SCO-240 is a potent, selective and oral somatostatin receptor subtype 5 (SSTR5) antagonist with IC50 of 2.0 nM (human SSTR5), >500-fold selectivity over other SSTR subtypes.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

SCO-240 is a potent, selective and oral somatostatin receptor subtype 5 (SSTR5) antagonist with IC50 of 2.0 nM (human SSTR5), >500-fold selectivity over other SSTR subtypes.

Physicochemical Properties

M.Wt 585.72
Formula C35H40FN3O4
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

6-(1-((2-cyclopropyl-5-ethoxy-4'-fluoro-[1,1'-biphenyl]-4-yl)methyl)piperidin-4-yl)-5-oxo-2-propyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carboxylic acid

References

1. Nishizaki H, et al. Clin Pharmacol Ther. 2024 Jun;115(6):1326-1335.

2. Patent WO/2015/052910.

3. Nishizaki H, et al. Eur J Endocrinol. 2026 May 7:lvag081.

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