SJ995973

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Chemical Structure : SJ995973

CAS No.: 2882065-25-8

Catalog No.: PC-23842Not For Human Use, Lab Use Only.

SJ995973 is a highly potent PROTAC degrader of bromodomain and extra-terminal (BET) proteins with DC50 of 0.87 nM in MV4-11 cells (BRD4) and Dmax=99%, inhibits viability of MV4-11 cells with IC50 of 3 pM.

Packing	Price	Stock
2 mg	$198	In stock
5 mg	$328	In stock
10 mg	$528	In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Physicochemical Properties

M.Wt	730.28
Formula	C37H40ClN7O5S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	2-((S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(5-(2-(4-(2,6-dioxopiperidin-3-yl)phenoxy)acetamido)pentyl)acetamide

References

1. Min J, et al. Angew Chem Int Ed Engl. 2021 Dec 13;60(51):26663-26670.

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SJ995973

Biological Activity

Physicochemical Properties

References

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