SJPYT-306 | PXR antagonist | Probechem Biochemicals

Chemical Structure : SJPYT-306

SJPYT-306 (SJPYT306)

Catalog No.: PC-22400Not For Human Use, Lab Use Only.

SJPYT-306 is a potent, selective dual antagonist and inverse agonist of pregnane X receptor (PXR) with binding IC50 of 6 nM, inverse agonist and antagonist IC50 of 1 nM and 14 nM, respectively.

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Biological Activity

SJPYT-306 is a potent, selective dual antagonist and inverse agonist of pregnane X receptor (PXR) with binding IC50 of 6 nM, inverse agonist and antagonist IC50 of 1 nM and 14 nM, respectively.

Physicochemical Properties

M.Wt	480.61
Formula	C27H36N4O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-N-(5-(tert-butyl)-2-(pentan-2-yloxy)phenyl)-1-(2,5-dimethoxyphenyl)-5-methyl-1H-1,2,3-triazole-4-carboxamide

References

1. Yongtao Li, et al. J Med Chem. 2022 Dec 22;65(24):16829-16859.

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SJPYT-306 (SJPYT306)

Biological Activity

Physicochemical Properties

References

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