SJPYT-331 | PXR antagonist | Probechem Biochemicals

Chemical Structure : SJPYT-331

SJPYT-331 (SJPYT331)

Catalog No.: PC-22401Not For Human Use, Lab Use Only.

SJPYT-331 is a potent, selective pregnane X receptor (PXR) antagonist with binding IC50 of 3.6 nM, antagonistic IC50 of 7.1 nM.

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Biological Activity

SJPYT-331 is a potent, selective pregnane X receptor (PXR) antagonist with binding IC50 of 3.6 nM, antagonistic IC50 of 7.1 nM.
SJPYT-331 blocks agonist-induced PXR activation in primary human hepatocytes (PHH).

Physicochemical Properties

M.Wt	496.56
Formula	C26H32N4O6
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	methyl (S)-3-(1-(2,5-dimethoxyphenyl)-5-methyl-1H-1,2,3-triazole-4-carboxamido)-4-(hexan-3-yloxy)benzoate

References

1. Garcia-Maldonado E, et al. Nat Commun. 2024 May 14;15(1):4054.

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SJPYT-331 (SJPYT331)

Biological Activity

Physicochemical Properties

References

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