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SR16435

Chemical Structure : SR16435

CAS No.: 857262-16-9

SR16435 (SR-16435)

Catalog No.: PC-61536Not For Human Use, Lab Use Only.

SR16435 is a mixed NOP/μ-opioid partial agonist with equally high affinity (Ki=29 nM) for both NOP and μ-opioid receptors.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    SR16435 is a mixed NOP/μ-opioid partial agonist with equally high affinity (Ki=29 nM) for both NOP and μ-opioid receptors.
    SR16435 possesses analgesic activity with reduced tolerance development and diminished reward in mice.

    Physicochemical Properties

    M.Wt 338.495
    Formula C22H30N2O
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    1-(1-(bicyclo[3.3.1]nonan-9-yl)piperidin-4-yl)indolin-2-one

    References

    1. Khroyan TV, et al. J Pharmacol Exp Ther. 2007 Feb;320(2):934-43.

    2. Zaveri NT, et al. J Med Chem. 2004 Jun 3;47(12):2973-6.

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