You are here:Home-Chemical Inhibitors & Agonists-GPCR-Adrenergic Receptor-SR59230A
SR59230A

Chemical Structure : SR59230A

CAS No.: 174689-39-5

SR59230A (SR-59230A)

Catalog No.: PC-22239Not For Human Use, Lab Use Only.

SR59230A is a potent, selective, and blood-brain barrier penetrating β3-adrenergic receptor antagonist with IC50 of 40, 408, and 648 nM for β3, β1, and β2 receptors, respectively.

Packing Price Stock Quantity
5 mg $98 In stock
10 mg $138 In stock
25 mg $248 In stock
50 mg $398 In stock
100 mg Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

SR59230A is a potent, selective, and blood-brain barrier penetrating β3-adrenergic receptor antagonist with IC50 of 40, 408, and 648 nM for β3, β1, and β2 receptors, respectively.

Physicochemical Properties

M.Wt 389.48
Formula C21H19N5OS
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

N-(2-aminophenyl)-4-[1-(2-thiophen-3-ylethyl)-1H-[1],[2],[3]triazol-4-yl]benzamide

References

1. Nisoli E, et al. Mol Pharmacol. 1996 Jan;49(1):7-14.

2. Manara L, et al. Br J Pharmacol. 1996 Feb;117(3):435-442.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: