SRX-246 | V1a receptor antagonist | Probechem Biochemicals

Chemical Structure : SRX-246

Catalog No.: PC-21615Not For Human Use, Lab Use Only.

SRX-246 (SRX246) is a potent, selective and CNS penetrant human V1a receptor antagonist with Ki of 0.3 nM.

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Biological Activity

SRX-246 (SRX246) is a potent, selective and CNS penetrant human V1a receptor antagonist with Ki of 0.3 nM.

M.Wt	703.88
Formula	C42H49N5O5
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-4-([1,4'-bipiperidin]-1'-yl)-4-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-N-((R)-1-phenylethyl)butanamide

1. Lago TR, et al. Psychopharmacology (Berl). 2021 Sep;238(9):2393-2403.

2. Fabio K, et al. Bioorg Med Chem. 2012 Feb 1;20(3):1337-45.

3. Guillon C, et al. Bioorg Med Chem. 2007;15:2054.