SSTR5 antagonist 1

Chemical Structure : SSTR5 antagonist 1

CAS No.: 1628741-91-2

Catalog No.: PC-26010Not For Human Use, Lab Use Only.

SSTR5 antagonist 1 (Compound 25a) is a selective and orally available somatostatin receptor subtype 5 (SSTR5) antagonist with IC50s of 9.6 and 57 nM for hSSTR5 and mSSTR5, respectively.

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5 mg	$248	In stock
10 mg	$398	In stock
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Biological Activity

SSTR5 antagonist 1 (Compound 25a) is a selective and orally available somatostatin receptor subtype 5 (SSTR5) antagonist with IC50s of 9.6 and 57 nM for hSSTR5 and mSSTR5, respectively.

Physicochemical Properties

M.Wt	511.59
Formula	C28H34FN3O5
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	1-(2-((2,6-Diethoxy-4'-fluoro-[1,1'-biphenyl]-4-yl)methyl)-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl)piperidine-4-carboxylic acid

References

1. Hirose H, et al. Bioorg Med Chem. 2017 Aug 1;25(15):4175-4193.

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