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Sarpogrelate hydrochloride

Chemical Structure : Sarpogrelate hydrochloride

CAS No.: 135159-51-2

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Sarpogrelate hydrochloride (MCI 9042;MCI9042;MCI-9042)

Catalog No.: PC-42655Not For Human Use, Lab Use Only.

A potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A.

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100 mg $256 In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

A potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A; also shows binding affinity for 5-HT2B; displays selectivity over 5-HT1-like, 5-HT3, beta, H1, H2 and M3; blocks serotonin-induced platelet aggregation.

Heart Failure

Approved

Physicochemical Properties

M.Wt 465.967
Formula C24H32ClNO6
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

DMSO: ≥ 62 mg/mL
Chemical Name/SMILES

Butanedioic acid, 1-[2-(dimethylamino)-1-[[2-[2-(3-methoxyphenyl)ethyl]phenoxy]methyl]ethyl] ester, hydrochloride (1:1)

References

1. Kikumoto R, et al. J Med Chem. 1990 Jun;33(6):1818-23.

2. Pertz H, et al. J Pharm Pharmacol. 1995 Apr;47(4):310-6.

3. Nishio H, et al. Arch Int Pharmacodyn Ther. 1996 Mar-Apr;331(2):189-202.

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