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Senktide

Chemical Structure : Senktide

CAS No.: 106128-89-6

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Senktide (NK3R antagonist)

Catalog No.: PC-63134Not For Human Use, Lab Use Only.

Senktide is a potent, selective agonist of neuromedin K3 (NK3) receptor (EC50 =0.5-3 nM), less potently agonizes the NK1 receptor (EC50=35 µM) and is without effect on the NK2 receptor.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Senktide is a potent, selective agonist of neuromedin K3 (NK3) receptor (EC50 =0.5-3 nM), less potently agonizes the NK1 receptor (EC50=35 µM) and is without effect on the NK2 receptor.

Physicochemical Properties

M.Wt 841.978
Formula C40H55N7O11S
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

DFFGLM (Modifications: Asp-1 = Succinyl-Asp, Phe-3 = Me-Phe, Met-6 = C-terminal amide)

References

1. Byk G, et al. J Med Chem. 1996 Aug 2;39(16):3174-8.

2. Sarau HM, et al. J Pharmacol Exp Ther. 1997 Jun;281(3):1303-11.

3. Harrison T, et al. Bioorg Med Chem Lett. 1998 Jun 2;8(11):1343-8.

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