Src Inhibitor 1 |CAS:179248-59-0 Probechem Biochemicals

Chemical Structure : Src Inhibitor 1

CAS No.: 179248-59-0

Src Inhibitor 1 (Src Kinase Inhibitor 1;Src-l1)

Catalog No.: PC-42303Not For Human Use, Lab Use Only.

A potent, selective dual site inhibitor of Src tyrosine kinase with Ki of 15 nM.

Packing	Price	Stock
5 mg	$56	In stock
10 mg	$76	In stock
25 mg	$176	In stock
50 mg	$316	In stock

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Biological Activity

A potent, selective dual site inhibitor of Src tyrosine kinase with Ki of 15 nM; has IC50 of 44 nM and 88 nM for Src and Lck, respectively; shows selectivity over VEGFR2 (88-fold) and C-fms (190-fold), also inhibits Csk and Yes with similar potency as Src, no activity against p38α/p38β MAPKs or CK1δ.

Physicochemical Properties

M.Wt	373.40456
Formula	C22H19N3O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	DMSO: 6.2 mg/mL (Need ultrasonic)
Chemical Name/SMILES	4-Quinazolinamine, 6,7-dimethoxy-N-(4-phenoxyphenyl)-

References

1. Tian G, et al. Biochemistry. 2001 Jun 19;40(24):7084-91.

2. Bain J, et al. Biochem J. 2007 Dec 15;408(3):297-315.

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Src Inhibitor 1 (Src Kinase Inhibitor 1;Src-l1)

Biological Activity

Physicochemical Properties

References

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