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TAK-802 hydrochloride

Chemical Structure : TAK-802 hydrochloride

CAS No.: 263248-36-8

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TAK-802 hydrochloride (TAK 802, TAK802)

Catalog No.: PC-61036Not For Human Use, Lab Use Only.

TAK-802 hydrochloride is a potent acetylcholinesterase (AChE) inhibitor with IC50 of 1.3 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    TAK-802 hydrochloride is a potent acetylcholinesterase (AChE) inhibitor with IC50 of 1.3 nM.
    TAK-802 exhibits high selectivity for acetylcholinesterase inhibition over butyrylcholinesterase inhibition.
    TAK-802 increases rhythmic bladder contractions in Guinea pigs and rats without affecting the basal intravesical pressure.

    Physicochemical Properties

    M.Wt 456.986
    Formula C26H30ClFN2O2
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    8-[3-[1-[(3-fluorophenyl)methyl]-4-piperidinyl]-1-oxopropyl]-1,2,5,6-tetrahydro-4H-pyrrolo[3,2,1-ij]quinolin-4-one hydrochloride

    References

    1. Ishichi Y, et al. Bioorg Med Chem. 2005 Mar 15;13(6):1901-11.

    2. Nagabukuro H, et al. Eur J Pharmacol. 2004 Feb 6;485(1-3):299-305.

    3. Nagabukuro H, et al. Eur J Pharmacol. 2004 Jun 28;494(2-3):225-32.

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