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TAS2R14 agonist 28.1

Chemical Structure : TAS2R14 agonist 28.1

CAS No.: 2883007-69-8

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TAS2R14 agonist 28.1 (Cmpd28.1, Compound 28.1)

Catalog No.: PC-20067Not For Human Use, Lab Use Only.

TAS2R14 agonist 28.1 is a potent, selective agonist of bitter taste receptor TAS2R14 with EC50 of 71 nM and Emax of 129%.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    TAS2R14 agonist 28.1 is a potent, selective agonist of bitter taste receptor TAS2R14 with EC50 of 71 nM and Emax of 129%.
    TAS2R14 agonist 28.1 shows a six-fold higher potency than flufenamic acid.
    TAS2R14 agonist 28.1 displays marked selectivity over a panel of 24 non-bitter taste human G protein-coupled receptors.

    Physicochemical Properties

    M.Wt 321.27
    Formula C13H10F3N7
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    N-(2-(1H-tetrazol-5-yl)phenyl)-4-methyl-6-(trifluoromethyl)pyrimidin-2-amine

    References

    1. Lukas Waterloo, et al. J Med Chem. 2023 Feb 27. doi: 10.1021/acs.jmedchem.2c01997.

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