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TASP0434299

Chemical Structure : TASP0434299

CAS No.: 1520893-08-6

TASP0434299 (TASP 0434299)

Catalog No.: PC-61507Not For Human Use, Lab Use Only.

TASP0434299 is a radioligand candidate for arginine vasopressin 1B (V1B) receptor that exhibits high binding affinities for human and rat V1B receptors with IC50 of 0.526 and 0.641 nM, respectively.

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    Biological Activity

    TASP0434299 is a radioligand candidate for arginine vasopressin 1B (V1B) receptor that exhibits high binding affinities for human and rat V1B receptors with IC50 of 0.526 and 0.641 nM, respectively.
    TASP0434299 shows no apparent binding affinities for other molecules at 1 uM.

    Physicochemical Properties

    M.Wt 509.607
    Formula C27H35N5O5
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    N-tert-butyl-2-[2-(3-methoxyphenyl)-6-[3-(morpholin-4-yl)propoxy]-4-oxopyrido[2,3-d]pyrimidin-3(4H)-yl]acetamide

    References

    1. Koga K, et al. J Pharmacol Exp Ther. 2016 Jun;357(3):495-508.

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