TC-N1752 | NaV1.7 inhibitor | Probechem Biochemicals

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Chemical Structure : TC-N1752

CAS No.: 1211866-85-1

TC-N1752 (TC-N 1752)

Catalog No.: PC-27183Not For Human Use, Lab Use Only.

TC-N1752 is a potent, state-dependent and orally active inhibitor of voltage gated sodium channel Nav1.7 with IC50 of 0.17 uM, 0.3 uM, 0.4 uM, 1.1 uM and 2.2 uM for hNav1.7, hNav1.3, hNav1.4, hNaV1.5 and rNav1.8, respectively, displays analgesic efficacy in the formalin pain model.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Physicochemical Properties

M.Wt	516.53
Formula	C25H27F3N6O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(2-Methyl-3-((4-(4-((4-(trifluoromethoxy)benzyl)oxy)piperidin-1-yl)-1,3,5-triazin-2-yl)amino)phenyl)acetamide

References

1. Howard Bregman, et al. J Med Chem. 2011 Jul 14;54(13):4427-45.

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TC-N1752 (TC-N 1752)

Biological Activity

Physicochemical Properties

References

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