TCPOBOP | CAR agonist | Probechem Biochemicals

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Chemical Structure : TCPOBOP

CAS No.: 76150-91-9

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TCPOBOP (CAR agonist)

Catalog No.: PC-49718Not For Human Use, Lab Use Only.

TCPOBOP is a phenobarbital-like class of CYP-inducing agent and agonist ligand for constitutive androstane receptor (CAR) with EC50 of 20 nM.

Packing	Price	Stock
10 mg	$78	In stock
25 mg	$128	In stock
50 mg	$198	In stock
100 mg	$298	In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

TCPOBOP is a phenobarbital-like class of CYP-inducing agent and agonist ligand for constitutive androstane receptor (CAR) with EC50 of 20 nM.
TCPOBOP competes directly for occupancy of the CAR LBD.
TCPOBOP enhances CAR interaction with the coactivator SRC-1 in vivo and in vitro.

Physicochemical Properties

M.Wt	402.05
Formula	C16H8Cl4N2O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1,4-bis((3,5-dichloropyridin-2-yl)oxy)benzene

References

1. Wei P, et al. Nature. 2000 Oct 19;407(6806):920-3.

2. Tzameli I, et al. Mol Cell Biol. 2000 May;20(9):2951-8.

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TCPOBOP (CAR agonist)

Biological Activity

Physicochemical Properties

References

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