TDO2 inhibitor Cpd-1

Chemical Structure : TDO2 inhibitor Cpd-1

Catalog No.: PC-23417Not For Human Use, Lab Use Only.

TDO2 inhibitor Cpd-1 is a potent, selective small molecule inhibitor of the apo form of human TDO2 with IC50 of 327 nM in human TDO2 cellular assay utilizing SW48 cells.

Packing	Price	Stock	Quantity
50 mg		Get quote
100 mg		Get quote
250 mg		Get quote

Get Quotation Now

* Please select Quantity before adding items.

or Bulk Inquiry

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Biological Activity

TDO2 inhibitor Cpd-1 is a potent, selective small molecule inhibitor of the apo form of human TDO2 with IC50 of 327 nM in human TDO2 cellular assay utilizing SW48 cells.
TDO2 inhibitor Cpd-1 showed almost no inhibition of IDO1, with respective IC50 values of 5.7 µM.

Physicochemical Properties

M.Wt	532.64
Formula	C30H36N4O5
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	ethyl 9-(3-(2-propylphenyl)-1-(1-phenylethyl)ureido)-2-methoxy-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine-3-carboxylate

References

1. Lotz-Jenne C, et al. Sci Rep. 2024 Nov 14;14(1):27937.

Overnight Delivery
Fast & Safe Delivery Worldwide
Rewards Program

About Us

Our Services

Site Map

Join with Us
Product Use Citations

Pharmacological Glossary Abbreviations

Abbreviations

Quality Manual

Inquiry Form
How to Order

Terms & Conditions

Credit Card Payment

Shipping Rates & Policies

Privacy Policy
sales@probechem.com