TDO2 inhibitor Cpd-2

Chemical Structure : TDO2 inhibitor Cpd-2

Catalog No.: PC-23418Not For Human Use, Lab Use Only.

TDO2 inhibitor Cpd-2 is a potent, selective small molecule inhibitor of the apo form of human TDO2 with IC50 of 14.8 nM in human TDO2 cellular assay utilizing SW48 cells.

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Biological Activity

TDO2 inhibitor Cpd-2 is a potent, selective small molecule inhibitor of the apo form of human TDO2 with IC50 of 14.8 nM in human TDO2 cellular assay utilizing SW48 cells.
TDO2 inhibitor Cpd-1 showed almost no inhibition of IDO1, with respective IC50 values of 5.7 µM.

Physicochemical Properties

M.Wt	532.64
Formula	C30H36N4O5
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	ethyl 9-(3-(2-isopropylphenyl)-1-((S)-1-phenylethyl)ureido)-2-methoxy-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine-3-carboxylate

References

1. Lotz-Jenne C, et al. Sci Rep. 2024 Nov 14;14(1):27937.

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