TGX286 | p110β inhibitor | Probechem Biochemicals

Chemical Structure : TGX286

TGX286 (TGX-286)

Catalog No.: PC-20453Not For Human Use, Lab Use Only.

TGX286 is a potent, selective p110β inhibitor with IC50 of 7, 17 and 13 nM for p110β WT, p110β D862Q, and p110β E858H, respectively, >100-fold selectivity over p110α.

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Biological Activity

TGX286 is a potent, selective p110β inhibitor with IC50 of 7, 17 and 13 nM for p110β WT, p110β D862Q, and p110β E858H, respectively, >100-fold selectivity over p110α.

Physicochemical Properties

M.Wt	358.44
Formula	C23H22N2O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	6-methyl-8-(1-(phenylamino)ethyl)-2-(pyridin-4-yl)-4a,8a-dihydro-4H-chromen-4-one

References

1. Frazzetto M, et al. Biochem J. 2008 Sep 15;414(3):383-90.

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TGX286 (TGX-286)

Biological Activity

Physicochemical Properties

References

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