TMX-4116 | CK1α PROTAC | Probechem Biochemicals

Chemical Structure : TMX-4116

TMX-4116 (TMX4116)

Catalog No.: PC-20151Not For Human Use, Lab Use Only.

TMX-4116 (TMX4116) is a highly potent casein kinase 1α (CK1α) degrader with DC50 of <200 nM (CK1α) in MOLT4 cells, does not degrade PDE6D and IKZF1/IKZF3.

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Biological Activity

TMX-4116 (TMX4116) is a highly potent casein kinase 1α (CK1α) degrader with DC50 of <200 nM (CK1α) in MOLT4 cells, does not degrade PDE6D and IKZF1/IKZF3.

Physicochemical Properties

M.Wt	389.43
Formula	C17H19N5O4S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	3-[4-[4-Methoxy-5-(1-pyrrolidinylcarbonyl)-3-thienyl]-1H-1,2,3-triazol-1-yl]-2,6-piperidinedione

References

1. Mingxing Teng, et al. J Med Chem. 2022 Jan 13;65(1):747-756.

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TMX-4116 (TMX4116)

Biological Activity

Physicochemical Properties

References

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