Catalog No.: PC-26243Not For Human Use, Lab Use Only.
Thioperamide (MR-12842) is a potent, selective, orally available, brain penetrant inverse agonist / antagonist of histamine H3-receptor (H3R) with Ki of 4.3 nM for inhibition of [3H]histamine release, inhibits [3H]histamine synthesis of KI of 31 nM.
Thioperamide (MR-12842) is a potent, selective, orally available, brain penetrant inverse agonist / antagonist of histamine H3-receptor (H3R) with Ki of 4.3 nM for inhibition of [3H]histamine release, inhibits [3H]histamine synthesis of KI of 31 nM.
