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Chemical Structure : Tianeptinostat
Catalog No.: PC-35281Not For Human Use, Lab Use Only.
Tianeptinostat is a potent class I HDAC inhibitor with IC50 of 28, 33 and 51 nM for HDAC1, 2 and 3, respectively, also inhibits HDAC6 (IC50=1.6 nM) but not HDAC5 (IC50>80 uM).
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Tianeptinostat is a potent class I HDAC inhibitor with IC50 of 28, 33 and 51 nM for HDAC1, 2 and 3, respectively, also inhibits HDAC6 (IC50=1.6 nM) but not HDAC5 (IC50>80 uM).
Tianeptinostat has EC50 of 1.72 and 7.66 uM in H3K9ac and H4K12ac assays, respectively.
| M.Wt | 437.939 | |
| Formula | C20H24ClN3O4S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Zhao WN, et al. ACS Chem Neurosci. 2018 Jun 22. doi: 10.1021/acschemneuro.8b00116.
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