UR-Po563 | H2 receptor agonist | Probechem Biochemicals

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Chemical Structure : UR-Po563

UR-Po563 (UR-Po 563)

Catalog No.: PC-49736Not For Human Use, Lab Use Only.

UR-Po563 is a potent, selective H2 receptor agonist with pKi of 7.75, >400-fold selectivity over H1R/H3R/H4R.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

UR-Po563 is a potent, selective H2 receptor agonist with pKi of 7.75, >400-fold selectivity over H1R/H3R/H4R.
UR-Po563 increased force of contraction in left atrium from H2-TG mice with pEC50 values of 8.27.
UR-Po563 increased force of contraction in isolated human right atrial muscle strips.

Physicochemical Properties

M.Wt	360.48
Formula	C17H24N6OS
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	Urea, N-[[[3-(2-amino-4-methyl-5-thiazolyl)propyl]amino]iminomethyl]-N′-[(1R)-1-phenylethyl]-

References

1. Ulrich Gergs, et al. J Pharmacol Exp Ther. 2021 Nov;379(3):223-234.

2. Biselli S, et al. Eur J Med Chem 214:113190

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UR-Po563 (UR-Po 563)

Biological Activity

Physicochemical Properties

References

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