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Chemical Structure : UR-Po563
Catalog No.: PC-49736Not For Human Use, Lab Use Only.
UR-Po563 is a potent, selective H2 receptor agonist with pKi of 7.75, >400-fold selectivity over H1R/H3R/H4R.
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UR-Po563 is a potent, selective H2 receptor agonist with pKi of 7.75, >400-fold selectivity over H1R/H3R/H4R.
UR-Po563 increased force of contraction in left atrium from H2-TG mice with pEC50 values of 8.27.
UR-Po563 increased force of contraction in isolated human right atrial muscle strips.
| M.Wt | 360.48 | |
| Formula | C17H24N6OS | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Ulrich Gergs, et al. J Pharmacol Exp Ther. 2021 Nov;379(3):223-234.
2. Biselli S, et al. Eur J Med Chem 214:113190
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