VRK1/CK1-IN-1

Chemical Structure : VRK1/CK1-IN-1

Catalog No.: PC-26318Not For Human Use, Lab Use Only.

VRK1/CK1-IN-1 is a potent, dual inhibitor of Vaccinia-related kinase 1 (VRK1) and the δ and ε isoforms of casein kinase 1 (CK1) with Ki of 37.9 nM for VRK1, and IC50 of 17 nM and 15 nM for CK1δ and CK1ε, mimics the cellular outcomes of VRK1 depletion.

Packing	Price	Stock	Quantity
25 mg		Get quote
50 mg		Get quote
100 mg		Get quote

Get Quotation Now

* Please select Quantity before adding items.

or Bulk Inquiry

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Biological Activity

Physicochemical Properties

M.Wt	416.39
Formula	C19H18F2N6O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-2-((3,5-Difluoro-4-hydroxyphenyl)amino)-7,8-dimethyl-5-((3-methylisoxazol-5-yl)methyl)-7,8-dihydropteridin-6(5H)-one

References

1. Fernando H de Souza Gama, et al. J Med Chem. 2024 Jun 13;67(11):8609-8629.

Overnight Delivery
Fast & Safe Delivery Worldwide
Rewards Program

About Us

Our Services

Site Map

Join with Us
Product Use Citations

Pharmacological Glossary Abbreviations

Abbreviations

Quality Manual

Inquiry Form
How to Order

Terms & Conditions

Credit Card Payment

Shipping Rates & Policies

Privacy Policy
sales@probechem.com

VRK1/CK1-IN-1

Biological Activity

Physicochemical Properties

References

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

Get Quote

* Indicates a Required FieldYour information is safe with us.