VU0152099 |CAS:612514-42-8 Probechem Biochemicals

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Chemical Structure : VU0152099

CAS No.: 612514-42-8

VU0152099 (VU 0152099)

Catalog No.: PC-62161Not For Human Use, Lab Use Only.

VU0152099 is a potent, selective, CNS-penetrant positive allosteric modulator of M4 mAChR with EC50 of 403 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

VU0152099 is a potent, selective, CNS-penetrant positive allosteric modulator of M4 mAChR with EC50 of 403 nM.
VU0152099 shows no agonist activity but potentiates responses of M(4) to acetylcholine, and is devoid of activity at other mAChR subtypes or at a panel of other GPCRs.
VU0152099 reverses amphetamine-induced hyperlocomotion in rats.

Physicochemical Properties

M.Wt	355.412
Formula	C18H17N3O3S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	3-amino-N-(1,3-benzodioxol-5-ylmethyl)-4,6-dimethylthieno[5,4-b]pyridine-2-carboxamide

References

1. Brady AE, et al. J Pharmacol Exp Ther. 2008 Dec;327(3):941-53.

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VU0152099 (VU 0152099)

Biological Activity

Physicochemical Properties

References

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