VU0415248 | M1 mAChR antagonist | Probechem Biochemicals

Chemical Structure : VU0415248

VU0415248 (VU 0415248)

Catalog No.: PC-20508Not For Human Use, Lab Use Only.

VU0415248 is a highly selective antagonist of muscarinic acetylcholine receptor subtype 1 (M1 mAChR) with IC50 of 0.4 uM and 0.18 uM for hM1R and rM1R, respectively.

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Biological Activity

VU0415248 is a highly selective antagonist of muscarinic acetylcholine receptor subtype 1 (M1 mAChR) with IC50 of 0.4 uM and 0.18 uM for hM1R and rM1R, respectively.
VU0415248 shows very high selectivity for the M1 receptor over the M2–5 subtypes across all five human and rat receptors.

Physicochemical Properties

M.Wt	425.51
Formula	C21H23N5O3S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	O=S(C1=CC=CC2=C1C=CC=N2)(NCCC(N3CCN(C4=CC=NC=C4)CC3)=O)=O

References

1. Bruce J Melancon, et al. Bioorg Med Chem Lett. 2012 Jan 15;22(2):1044-8.

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VU0415248 (VU 0415248)

Biological Activity

Physicochemical Properties

References

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