Chemical Structure : VU0453595
CAS No.:
1432436-13-9
VU0453595
(VU 0453595, VU-0453595, VU453595, VU595)
Catalog No. : PC-35478Not For Human Use, Lab Use Only.
VU0453595 (VU453595) is a potent, selective M1 positive allosteric modulator (PAM) with EC50 of 3.2 uM (rM1).
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-3547801
Biological Activity
VU0453595 (VU453595) is a potent, selective M1 positive allosteric modulator (PAM) with EC50 of 3.2 uM (rM1).
Physicochemical Properties
M.Wt
322.343
Formula
C18H15FN4O
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
6-[[2-Fluoro-4-(1-methyl-1H-pyrazol-4-yl)phenyl]methyl]-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-5-one
References
1. Ghoshal A, et al. Neuropsychopharmacology.
2. Panarese JD, et al. Bioorg Med Chem Lett.
3. Lv X, et al. Neuropharmacology.
4. Moran SP, et al. Neuropsychopharmacology.
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