Chemical Structure : VU0467485
CAS No.:
1451994-10-7
VU0467485
(VU-0467485;AZ13713945)
Catalog No. : PC-35946Not For Human Use, Lab Use Only.
VU0467485 (VU-0467485, AZ13713945) is potent, selective, and orally bioavailable muscarinic acetylcholine receptor 4 (M4) positive allosteric modulator with EC50 of 78.8 nM (hM4).
Packing Price Stock Quantity 5 mg $128 In stock 0 1 2 3 4 5 10 mg $188 In stock 0 1 2 3 4 5 25 mg $328 In stock 0 1 2 3 4 5 50 mg $528 In stock 0 1 2 3 4 5 100 mg Get quote 0 1 2 3 4 5
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-3594601
Biological Activity
VU0467485 (VU-0467485, AZ13713945) is potent, selective, and orally bioavailable muscarinic acetylcholine receptor 4 (M4 ) positive allosteric modulator with EC50 of 78.8 nM (hM4).
Physicochemical Properties
M.Wt
360.407
Formula
C17H17FN4O2S
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
5-amino-N-(3-fluoro-4-methoxybenzyl)-3,4-dimethylthieno[2,3-c]pyridazine-6-carboxamide
References
1. Wood MR, et al. ACS Med Chem Lett
2. Melancon BJ, et al. Bioorg Med Chem Lett
3. Deng X, et al. ChemMedChem
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